SEEK ID: https://fairdomhub.org/people/2256
Location:
Italy
ORCID:
https://orcid.org/0000-0003-2574-3911
Joined: 25th Oct 2022
Expertise: structural biology, Cancer research, parassite research, drug development, antibiotic resistance, drug resistance, antibacterial drugs, neurodegenerative diseases, metalloproteins, protein-protein interactions, protein production
Tools: X-ray crystallography, Protein chemical methods (protein overproduction, recombinant technology, recombinant protein production, Site-directed mutagenesis, Spectroscopy and structural analysis
Related items
The recent COVID19 pandemic infection has undisclosed long-standing issues in the translation of drugs from animals to humans or vice-versa. Nearly 75% of emerging human infections worldwide originated from animals; existing drugs for human and animal (H&A) vector-borne diseases (VBD) are scarce, with limited efficacy, toxicity, and finite resources. Emerging environmental problems in pharmaceutical use/manufacturing increase attention in the field. The two drug pipelines are developed ...
Projects: WG1 - Compound libraries coordination and integration of compound design, WG2 - Integration of early phase studies and low environmental impact actions, WG3 - Coordination of in vitro-to-in vivo translation of OneHealth leads and candidates, WG4 - Integration of R&D process-environmental studies and translation in informed whitepaper, WG5 - Promote dissemination, WG6 - Promote the transfer of knowledge, BioTarget Database, Compound Data
Web page: https://onehealthdrugs.com/
Public web page: Not specified
Public web page: Not specified
Organisms: Not specified
Public web page: Not specified
Organisms: Not specified
Public web page: Not specified
Organisms: Not specified
Public web page: Not specified
Organisms: Not specified
Public web page: Not specified
Organisms: Not specified
ROR ID: Not specified
Department: Not specified
Country:
Italy
City: Siena
Web page: https://www.unisi.it/
Abstract (Expand)
Authors: J. Panecka-Hofman, P. Linciano, I. Pohner, E. Dyguda-Kazimierowicz, W. Jedwabny, G. Landi, N. Santarem, G. Witt, B. Ellinger, M. Kuzikov, R. Luciani, S. Ferrari, D. Aiello, S. Mangani, C. Pozzi, A. Cordeiro-da-Silva, S. Gul, M. P. Costi, R. C. Wade
Date Published: 9th Oct 2025
Publication Type: Journal Article
PubMed ID: 41026998
Citation: J Med Chem. 2025 Oct 9;68(19):20595-20618. doi: 10.1021/acs.jmedchem.5c01799. Epub 2025 Sep 30.
Abstract
Authors: Valeria Francesconi, Marco Rizzo, Cecilia Pozzi, Lorenzo Tagliazucchi, Claude U. Konchie Simo, Giulia Saporito, Giacomo Landi, Stefano Mangani, Anna Carbone, Silvia Schenone, Nuno Santarém, Joana Tavares, Anabela Cordeiro-da-Silva, Maria Paola Costi, Michele Tonelli
Date Published: 2nd Jul 2024
Publication Type: Journal Article
DOI: 10.1021/acsinfecdis.4c00113
Citation: ACS Infect. Dis. 10(8):2755-2774.
Abstract
Authors: Pasquale Linciano, Cecilia Pozzi, Giusy Tassone, Giacomo Landi, Stefano Mangani, Matteo Santucci, Rosaria Luciani, Stefania Ferrari, Nuno Santarem, Lorenzo Tagliazucchi, Anabela Cordeiro-da-Silva, Michele Tonelli, Donatella Tondi, Laura Bertarini, Sheraz Gul, Gesa Witt, Carolina B. Moraes, Luca Costantino, Maria Paola Costi
Date Published: 2024
Publication Type: Journal Article
DOI: 10.1016/j.ejmech.2023.115946
Citation: European Journal of Medicinal Chemistry 264:115946.
Their tags